Inhibitor class | Agents | Potency IC50(nM) |
Pan-PI3K inhibitor | Pictilisib | PI3Kα/δ 3 |
Pan-PI3K inhibitor | Buparisib | PI3Kα 52PI3Kδ 116 PI3Kβ 166PI3Kγ 262 |
Pan-PI3K inhibitor | Copanlisib | PI3Kα 0.5PI3Kδ 0.7 PI3Kβ 3.7PI3Kγ 6.4 |
Isoform-Selective PI3K Inhibitors | Alpelisib | PI3Kα 5 |
Isoform-Selective PI3K Inhibitors | Taselisib | PI3Kα 0.29 |
Isoform-Selective PI3K Inhibitors | Idelalisib | p110δ 2.5 |
Dual PI3K/mTOR Inhibitors | Omipalisib | p110α 0.019 mTORC10.18 |