Inhibitor class

Agents

Potency IC50(nM)

Pan-PI3K inhibitor

Pictilisib

PI3Kα/δ 3

Pan-PI3K inhibitor

Buparisib

PI3Kα 52PI3Kδ 116

PI3Kβ 166PI3Kγ 262

Pan-PI3K inhibitor

Copanlisib

PI3Kα 0.5PI3Kδ 0.7

PI3Kβ 3.7PI3Kγ 6.4

Isoform-Selective PI3K Inhibitors

Alpelisib

PI3Kα 5

Isoform-Selective PI3K Inhibitors

Taselisib

PI3Kα 0.29

Isoform-Selective PI3K Inhibitors

Idelalisib

p110δ 2.5

Dual PI3K/mTOR Inhibitors

Omipalisib

p110α 0.019

mTORC10.18