Entry

R1

R2

产物

产率

1

H

p-CH3

3aa

76

2

p-CH3

p-CH3

3ab

72

3

p-F

p-CH3

3ac

70

4

o-CH3

p-CH3

3ad

55

5

o-Cl

p-CH3

3ae

trace

6

m-CH3

p-CH3

3af

56

7

H

p-OCH3

3ba

64

8

H

p-CF3

3bb

61

9

H

m-CH3

3bc

58