Entry | R1 | R2 | 产物 | 产率 |
1 | H | p-CH3 | 3aa | 76 |
2 | p-CH3 | p-CH3 | 3ab | 72 |
3 | p-F | p-CH3 | 3ac | 70 |
4 | o-CH3 | p-CH3 | 3ad | 55 |
5 | o-Cl | p-CH3 | 3ae | trace |
6 | m-CH3 | p-CH3 | 3af | 56 |
7 | H | p-OCH3 | 3ba | 64 |
8 | H | p-CF3 | 3bb | 61 |
9 | H | m-CH3 | 3bc | 58 |