Entry

R

Yieldsb (%)

m.p. (℃)

Found

Reported [lit.]

4a

C6H5

89

90~92

89~91 [15]

4b

4-Me-C6H4

75

116~118

118~120 [16]

4c

2-MeO-C6H4

82

68~69

66~68 [13]

4d

3-MeO-C6H4

80

116~117

113~115 [13]

4e

4-F-C6H4

81

103~105

105~107 [15]

4f

2-Cl-C6H4

80

139~140

136~138 [16]

4g

2-Br-C6H4

84

121~123

121~122 [10]

4h

2-NO2-C6H4

81

120~122

121~123 [16]