Entry

R

Yield [%]

Dr

ee [%]

1

5-H

89

17:1

99

2

5-Me

63

13:1

98

3

5-OMe

58

10:1

96

4

5-F

86

>20:1

98

5

5-Cl

92

>20:1

98

6

5-Br

94

>20:1

98

7

5-I

91

>20:1

97

8

5-NO2

98

>20:1

98

9

5-OCF3

92

>20:1

96

10

6-Cl

94

>20:1

97