| 化合物 | 结构式 | 适应症 | 公司 |
| 1 .Ibrutinib |
| MCL, CLL, SLL, WM, cGVHD, etc. | Pharmacyclics/Johnson |
| 2. Acalabrutinib |
| MCL, CLL, SLL | Acerta Pharma |
| 3. Zanubrutinib |
| MCL | BeiGene |
| 4. Tirabrutinib |
| PCNSL | Ono Pharma |
| 5. Orelabrutinib |
| MCL, CLL, SLL | InnoCare Pharma |